FAQ Categories Opioids

55. Concise Synthesis of GB22 by Endo-Selective Siloxycyclopropane Arylation

55. Burdge, H. E.; Oguma, T.; Kawajiri, T.; Shenvi, R. A. Concise Synthesis of GB22 by Endo-Selective Siloxycyclopropane Arylation ChemRxiv DOI: 10.26434/chemrxiv.8263415.v1 .

47. Intermolecular Heck Coupling with Hindered Alkenes Directed by Potassium Carboxylates

47. Huffman, T.; Wu, Y.; Emmerich, A.; Shenvi, R.A. Intermolecular Heck Coupling with Hindered Alkenes Directed by Potassium Carboxylates Angew. Chem. Int. Ed. 2019, 58, 2371-2376.

40. A Review of Salvinorin Analogs and their Kappa-Opioid Receptor Activity

40. Roach, J. J.; Shenvi, R. A. A Review of Salvinorin Analogs and their Kappa-Opioid Receptor Activity. Bioorg. Med. Chem. Lett. 2018, 28, 1436–1445. DOI: 10.1016/j.bmcl.2018.03.029

39. O6C-20-nor-SalA is a stable and potent KOR agonist

39. Hirasawa, S.; Cho, M.; Brust, T. F.; Roach, J. J.; Bohn, L. M.; Shenvi, R. A. O6C-20-nor-SalA is a stable and potent KOR agonist. Bioorg. Med. Chem. Lett. 2018, 28, 2770–2722. Special Issue dedicated to Dale Boger.

38. Dynamic Strategic Bond Analysis Yields a 10-step Synthesis of 20-nor-SalA, a Potent Κ-OR Agonist

38. Roach, J. J.; Sasano, Y.; Schmid, C. L.; Zaidi, S.; Katrich, V.; Stevens, R. C.; Bohn, L. M.; Shenvi, R. A. Dynamic Strategic Bond Analysis Yields a 10-step Synthesis of 20-nor-SalA, a Potent Κ-OR Agonist. A(CS)2 2017, 3, 1329–1336. ChemRxiv DOI: 10.26434/chemrxiv.5318188 #1 Most Viewed Article on ChemRxiv, Aug-Dec 2017. Highlighted by Tien Ngyuen in C&EN, Sept. [...]